Molecular Search Results
Search for: P21817 in all (Fuzzy Match)
Found 53 recordings
| DICL ID | Ion Channel | Compound Function | Species | Value | References | |
|---|---|---|---|---|---|---|
| DICL_CP_0350256 | Ryanodine receptor 1 | Inhibitor | Homo sapiens (Human) | IC50: 4200 nM | 10.1038/ja.2009.126, 20057513 | |
| DICL_CP_0373602 | Ryanodine receptor 1 | Blocker | Homo sapiens (Human) | IC50: 5100 nM | 10.1124/mol.109.057265, 19509218 | |
| DICL_CP_0398557 | Ryanodine receptor 1 | Agonist | Homo sapiens (Human) | EC50: 11000 nM | 10.1016/j.bmcl.2008.09.080, 18851910 | |
| DICL_CP_0402556 | Ryanodine receptor 1 | Activator | Homo sapiens (Human) | EC50: 14700 nM | 10.1021/np020382h, 12542356 | |
| DICL_CP_0416536 | Ryanodine receptor 1 | Inactive | Homo sapiens (Human) | Inhibition: No effect | 10.1124/mol.111.074740, 21989257 | |
| DICL_CP_0417415 | Ryanodine receptor 1 | Activator | Homo sapiens (Human) | EC50: 52000 nM | 10.1371/journal.pone.0054208, 23349825 | |
| DICL_CP_0418598 | Ryanodine receptor 1 | Inhibitor | Homo sapiens (Human) | IC50: 1.5 nM | US10538528 | |
| DICL_CP_0423842 | Ryanodine receptor 1 | Inhibitor | Homo sapiens (Human) | IC50: 1.7 nM | US10538528 | |
| DICL_CP_0426595 | Ryanodine receptor 1 | Antagonist | Homo sapiens (Human) | IC50: 3.5 nM | 10.1021/jm950711l, 8691427 | |
| DICL_CP_0426596 | Ryanodine receptor 1 | Antagonist | Homo sapiens (Human) | IC50: 3.3 nM | 10.1021/jm950711l, 8691427 |
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